DR ANTHONY MELVIN CRASTO,WorldDrugTracker, helping millions, A 90 % paralysed man in action for you, I am suffering from transverse mylitis and bound to a wheel chair,With death on the horizon, This will not stop me, Gods call only..........
DR ANTHONY MELVIN CRASTO Ph.D ( ICT, Mumbai) , INDIA 29Yrs Exp. in the feld of Organic Chemistry,Working for GLENMARK PHARMA at Navi Mumbai, INDIA. Serving chemists around the world. Helping them with websites on Chemistry.Million hits on google, world acclamation from industry, academia, drug authorities for websites, blogs and educational contributio
n

Monday 30 November 2015

Harold E Varmus






Harold Eliot Varmus is an American Nobel Prize-winning scientist and the 14th Director of the National Cancer Institute, a post to which he was appointed by President Barack Obama. He was a co-recipient of the 1989 Nobel Prize in Physiology or Medicine for discovery of the cellular origin of retroviraloncogenes. He also serves as one of three co-Chairs of thePresident's Council of Advisors on Science and Technology.









With Prof. Harold Varmus! 
smile emoticon — at Hebrew University of Jerusalem.







JERUSALEM ISRAEL

DRUG APPROVALS BY DR ANTHONY MELVIN CRASTO .....FOR BLOG HOME CLICK HERE


Join me on Linkedin

View Anthony Melvin Crasto Ph.D's profile on LinkedIn

Join me on Facebook FACEBOOK
Join me on twitterFollow amcrasto on Twitter     
Join me on google plus Googleplus

 amcrasto@gmail.com

/////////

Dr. Sandeep N. Raikar

.

 Dr. Sandeep N. Raikar
Dr. Sandeep N. Raikar did his BSc and MSc from Sri Satya Sai Institute of Higher Learning-India. He then moved to University of Kansas where he worked with Prof. Helena C. Malinakova and obtained his Ph.D. degree in 2013. Currently he is a postdoctoral associate in Prof. Huw M. L. Davies laboratory at Emory University.
////////////






 DRUG APPROVALS BY DR ANTHONY MELVIN CRASTO .....FOR BLOG HOME CLICK HERE


Join me on Linkedin

View Anthony Melvin Crasto Ph.D's profile on LinkedIn

Join me on Facebook FACEBOOK
Join me on twitterFollow amcrasto on Twitter     
Join me on google plus Googleplus

 amcrasto@gmail.com


Jin-Quan Yu

.
 Jin-Quan Yu


Jin-Quan Yu received his BSc in Chemistry from East China Normal University and his MSc from the Guangzhou Institute of Chemistry. In 2000, he obtained his PhD at the University of Cambridge with Prof. J. B. Spencer. Following time as a junior research fellow at Cambridge, he joined the laboratory of Prof. E. J. Corey at Harvard University as a postdoctoral fellow. He then began his independent career at Cambridge (2003-2004), before moving to Brandeis University (2004-2007), and finally to The Scripps Research Institute, where he is currently Frank and Bertha Hupp Professor of Chemistry. His group studies transition metal-catalyzed C-H activation.

 Department of Chemistry, The Scripps Research Institute (TSRI), 10550 N. Torrey Pines Road, La Jolla, CA 92037 (USA). E-mail: yu200@scripps.edu.








/////////////

Keary Mark Engle

.

Keary Mark Engle


  Keary Mark Engle graduated Phi Beta Kappa and summa cum laude from the University of Michigan, where he worked with Prof. Adam Matzger studying self-assembled monolayers. A Fulbright Scholar, he spent the 2007-2008 academic year studying under the tutelage of Prof. Manfred Reetz at the Max-Planck-Institut für Kohlenforschung (Germany). He completed his graduate work jointly at The Scripps Research Institute and the University of Oxford, under the supervision of Prof. Jin-Quan Yu and Prof. Véronique Gouverneur, respectively, earning a Ph.D. in Chemistry and a DPhil in Biochemistry. During graduate school, his honors included NSF and NDSEG Predoctoral Fellowships. Presently, Keary is an NIH Postdoctoral Fellow with Prof. Robert H. Grubbs at Caltech.









//////////

Dong-Hui Wang

.

 Dong-Hui Wang


 Dong-Hui Wang completed his BSc at Lanzhou University in 2000 then carried out research at the Shanghai Institute of Organic Chemistry under Prof. Zhaoguo Zhang. In 2004, he began graduate studies under Prof. Jin-Quan Yu. He earned his MSc from Brandeis University before relocating to The Scripps Research Institute, where he completed his Ph.D. in 2010. His thesis research was recognized with the Chinese Government Award for Outstanding Self-Financed Students Abroad. Dong-Hui worked as a postdoctoral research fellow in the laboratory of Prof. Stephen Buchwald at MIT (2010-2012), and as a medicinal chemist at Abide Therapeutics (2012-2014). Presently, he is an Assistant Professor at the Shanghai Institute of Organic Chemistry (China).










////////////

Yutaka Kobayashi



Yutaka Kobayashi

Yutaka Kobayashi received a B.S. in chemistry from Kitasato University in 2008. He received a Ph.D. in Life Sciences from Kitasato University under the guidance of Professor Toshiaki Sunazuka. He is currently a post-doctoral fellow in the laboratory of Professor John L. Wood at Baylor University.

Yu-Pu Wang

Yu-Pu Wang


Yu-Pu Wang was born in Taipei, Taiwan. He received a B.S. degree in Chemistry in 2009 from Rice University working in the laboratory of Professor James M. Tour. He is currently pursuing a Ph.D. degree at the Massachusetts Institute of Technology in the research group of Professor Rick L. Danheiser and his work involves the development of new methods for the synthesis of highly substituted indoles and their application to the synthesis of natural products and polycyclic systems with interesting electronic properties.

James Deng

James Deng


James Deng was born in New Haven, Connecticut and is currently an undergraduate chemistry major at the Massachusetts Institute of Technology and is expecting to graduate with a B.S. degree in chemistry in 2017. James joined the laboratory of Professor Danheiser as an undergraduate researcher in January 2014 and is currently investigating a synthetic route to bioactive polyacetylene natural products.

Rick L. Danheiser

.
 Rick L. Danheiser




Rick L. Danheiser received his undergraduate education at Columbia where he carried out research in the laboratory of Professor Gilbert Stork. He received his Ph.D. at Harvard in 1978 working under the direction of E. J. Corey on the total synthesis of gibberellic acid. Dr. Danheiser is the A. C. Cope Professor of Chemistry at MIT where his research focuses on the design and invention of new annulation and cycloaddition reactions, and their application in the total synthesis of biologically active compounds.

Pauline van Meurs

Pauline van Meurs.

 Pauline van Meurs




Experience

Group Leader

Mercachem
– Present (10 years 9 months)
Responsible for the day-to-day supervision of assigned team members.
Responsible for the progress of my own projects and projects performed by the project team. This includes planning, syntheses, literature research, quote calculations, reporting, shipment tracking, post-calculation, databases, hours registration and communication to the customer.
Responsible for the day-to-day operations at the laboratory.

Research Scientist

Mercachem
(2 years 4 months)
Perform all common organic preparative laboratory work
Guidance of research chemists (HLO-ers)

PhD

Eindhoven University of Technology
(4 years 3 months)
PhD research in the Group Supramolecular and Macromolecular Organic Chemistry of Prof. Dr. Ir. R. A. J. Janssen en Prof. Dr. E. W. Meijer.
Titel thesis: High-spin molecules of p-phenylenediamine radical cations.
The search for an organic material that exhibits magnetic properties is a scientific challenge. The research described in the thesis is focused on the design, synthesis, and characterization of organic molecules, which, upon doping, have multiple unpaired electrons that exhibit intra- or intermolecular ferromagnetic coupling resulting in high-spin molecules and architectures.





Education

Leiden University

MsC, Chemistry

CLA

 Map of eindhoven university of technology
//////////

Sunday 29 November 2015

Fredrik Tinnis

Fredrik Tinnis

Fredrik Tinnis obtained his Ph.D. degree from Stockholm University (2014) under the supervision of Prof. Hans Adolfsson, where he focused on the development of catalytic procedures for the formation of amides. Fredrik is now a post-doctoral fellow in the same research group and is currently working on chemoselective reduction of amides.

Education

Experience

Postdoctoral Researcher

Stockholm University
– Present (1 year 5 months)

Research Assistant

Stockholm University
(3 months)

PhD Student

Stockholm University
(5 years)Stockholm, Sweden

Accounting Manager

FDS Financial Distribution Serivices AB
(5 years 1 month)Stockholm, Sweden

Head of Administration

FDS Financial Distribution Services AB
(5 years 1 month)
 

 https://www.researchgate.net/profile/Fredrik_Tinnis
 https://www.researchgate.net/profile/Fredrik_Tinnis/contributions
https://www.linkedin.com/in/fredrik-tinnis-6a938170



Research Experience

  • Jun 2014–
    present
    PostDoc Position
    Stockholm University · Department of Organic Chemistry · Prof. Hans Adolfsson
    Sweden · Stockholm
  • Aug 2013–
    present
    PhD Student
    Stockholm University · Department of Organic Chemistry
    Sweden · Stockholm

Education

  • Aug 2004–
    Jun 2009
    Stockholm University
    Organic chemistry · Master
    Sweden · Stockholm



From left to right: Helena Lundberg, Fredrik Tinnis, Dr Nicklas Selander, and Professor Hans Adolfsson



//////////

Friday 27 November 2015

Dr. Santosh J. Gharpure





Dr. Santosh J. Gharpure
Associate professor,
Department of Chemistry,
Indian Institute of Bombay,
Powai, Mumbai-400076.



Work Tel: (022) 2576 7171
Home Tel: (022) 2576 817

E-mail: sjgharpure@iitb.ac.in

sjgharpure[at]chem.iitb.ac.in sjgharpure[at]iitb.ac.in

http://www.chem.iitb.ac.in/~sjgharpure/gallery.html

http://www.chem.iitb.ac.in/~sjgharpure/images/sjg-cv.pdf

http://www.chem.iitb.ac.in/people/Faculty/prof/sjg.html

https://www.researchgate.net/profile/Santosh_Gharpure

https://in.linkedin.com/in/santosh-gharpure-90398711

 

 

 

Dr. Santosh J. Gharpure graduated with an M.Sc. degree in 1996, from Indian Institute of Technology Bombay, Powai. He obtained Ph.D. from Indian Institute of Science, Bangalore working with Late Prof. A. Srikrishna in 2001. He held a post-doctoral position with Prof. P. Andrew Evans at Indiana University, Bloomington, U.S.A. Subsequently; he joined the Department of Chemistry, IIT Madras, Chennai in the year 2004. In 2012, he moved to Department of Chemistry, IIT Bombay, Powai, Mumbai as an associate professor. His research focuses on organic chemistry pertaining to natural and unnatural product synthesis and developing new synthetic methodologies.

Dr. Gharpure is a recipient of INSA Medal for Young Scientist. He was awarded IIT Madras Young Faculty Recognition Award (YFRA) for his contribution in teaching and research in 2010. He received B. M. Birla science Prize in Chemistry for the year 2011. Recently, he was selected as one of the Thieme Chemistry Journal Awardees for the year 2013.

 

 

 

Our broad areas of Research Interests include :

  • Organic synthesis
  • New synthetic methods
  • Asymmetric synthesis
  • Natural product synthesis
  • Catalysis
  • Organometallic chemistry

Education :

View CV in pdf form :
Degree University/Institute Year
Ph.D IISc, Bangalore (Ph.D. in Synthetic Organic Chemistry with Professor A. Srikrishna, "Enantiospecific Approaches to Neopupukeananes") Aug 1996 - July 2001
M.Sc. IIT Bombay, (M.Sc. in Organic Chemistry, M.Sc. Project with Professor S. V. Bhat, "Synthesis and Evaluation of Biological Activity of Polyenes") July 1994 - April 1996
B.Sc. V. G. Vaze College, University of Bombay, Mumbai July 1989 - June 1994

Professional Experience :

Employment University/Institute Year
Post-Doctoral Fellow with Professor P. Andrew Evans Dept. of Chemistry, Indiana University, Bloomington Aug 2001 - April 2004
Assistant Professor IIT Madras May 2004 - July 2012
Associate Professor IIT Bombay July 2012 - present

Honors and Awards :

KET's V. G. Vaze Alumni Achievers Award, January 2013.
Selection as one of the Thieme Chemistry Journal Awardees 2013, December 2012.
B.M. Birla Science Prize in Chemistry, November 2012.
Awarded Young Faculty Recognition Award (YFRA) by IIT Madras, Chennai, September 2010.
Awarded INSA Medal for Young Scientist by Indian National Science Academy, New Delhi, India, April 2008.
Junior and Senior Research Fellow of Council for Scientific and Industrial Research, New Delhi, India, Aug. 1996-July 2001.
Qualified Graduate Aptitude Test in Engineering, All India Rank-1, March 1996.
Winner of the Gold Medal at the Chemistry Aptitude Test held by the Indian Chemical Society, March 1995.
17th Rank in the Merit List of the S.S.C. Board Examination Held by Maharashtra Board, July 1989.

Memberships :

Chemical Research Society of India (CRSI)
American Chemical Society (ACS)
Indian Association of Chemistry Teachers (IACT)
 avatar for Santosh Gharpure

Research :


In the broad area of Organic Chemistry, the main focus of Prof. Gharpure's research has been the development of new synthentic methods, which would be applicable for the synthesis of natural and unnatural products of biological relevance.


Synthetic Methodology :

We have used vinylogous functional groups, namely vinylogous carbonate and carbamate, in the stereoselective synthesis of oxa- and aza-cycles. The reactivity of vinylogous carbonates/carbamates was studied under a variety of conditions. Thus, our group has used radical cyclisation to vinylogous carbonates/carbamates for the stereoselective synthesis of new oxa-cages as well as angular oxa- and aza-triquinanes. An efficient strategy for the synthesis of tetrahydrofurans (THFs), tetrahydropyrans (THPs) and oxepane derivatives has been developed employing a tandem SN2-Michael addition to vinylogous carbonates. On the other hand, intramolecular cyclopropanation of vinylogous carbonates/carbamates using carbenes led to the oxygen and nitrogen bearing donor-acceptor substituted cyclopropanes (DACs). These DACs could be converted into diversely functionalized THFs, THPs, lactones, pyrrolidine, piperidine and lactam derivatives, which is again explored for the total synthesis of bioactive molecules such as butanolide and butenolide based natural products.Vinylogous carbonates/carbamates were also found to give useful reactions in the presence of Lewis acids undergoing intramolecular Pictet-Spengler as well as Prins type cyclizations leading to N-fused oxazinoindoles, dihydrobenzofurans and dihydroindole derivatives.



Natural Product Synthesis :

Apart from using vinylogous functional groups in the synthesis of oxa- and aza-cycles, our group has developed efficient strategies for the synthesis of flavans and isoflavans. Flavans and isoflavans are class of compounds, which are thought to be responsible for biological activity of traditional Chinese medicines. The strategy relying on o-quinone methides has been used for the total synthesis of variety of natural products of this family like equol, 3'-hydroxyequol, vestitol and myristinins.






Very recently, we have also developed stereoselective strategies for construction of morpholines and oxazepenes, which are important pharmacophores.This method also used for the total synthesis of chelonin A and Chelonin C. 

Research Highlights :

  1. "Shortest Route to Mucocin", C & E News2003, 81(49), 32.

  2. "Synthesis of Heterocyclic Triquinanes via Sequential Radical Cyclizations", Victor Snieckus and Nathan E. Genung (Pfizer), Synfacts2013, 9, 33.

  3. "Young Career Focus: Dr. Santosh J. Gharpure (Indian Institute of Technology Bombay, Mumbai, India)", Synstories, SYNFORM, 2014/03, Published online: 17.02.2014, DOI: 10.1055/s-0033-1340792.






Publications :




Current Work :


48. Counter Ion Dependent Alkyne Iminium Ion Cyclization for Divergent Synthesis of N-Fused Indolylidine, Indole and Indoline Derivatives Promoted by the Lewis/Bronsted Acid.
S. J. Gharpure, Y. G. Shelke and D. P. Kumar, Org. Lett. accepted.



47. Stereoselective Synthesis of cis-2,6-DisubstitutedMorpholines and 1,4-Oxathianes by Intramolecular Reductive Etherification of 1,5-Diketones.
S. J.Gharpure, D. Anuradha, J. V. K Prasad, and P. S. Rao, Eur. J. Org. Chem., 2015, 86-90.



46.Donor-Acceptor Substituted Cyclopropane to Butanolide and Butenolide Natural Products: Enantiospecific First Total Synthesis of (+)-Hydroxyancepsenolide.
S. J. Gharpure, Laxmi Narayan Nanda and M. K. Sukla, Org. Lett.2014,16, 6424?6427.



45.On the Photophysics of ButadiyneBridged Pyrene-Phenyl Molecular Conjugates: Multiple Emissive Pathways Through Locally Excited, Intramolecular Charge Transfer and ExcimerStates.
A. K.Pati, S. J. Gharpure and A. K. Mishra,Faraday Discuss.2014.(Invited)


44.Synthesis of IsochromeneDerivatives using an Intramolecular Benzylic C(sp3)-C(sp2) Bond Forming Heck Reaction on Vinylogous Carbonates.
S.J. Gharpure ,Yogesh, G. Shelke and S.R.B. Reddy,RSC Adv.,2014, 4, 46962-46965.



43. Stereoselective Synthesis of C-fused Pyranoindoles, Pyranobenzofurans and PyranobenzothiopheneScaffolds using Oxa-Pictet-Spengler Type Teaction of Vinylogous Carbonates.
S. J. Gharpure and V. Prasath,Org. Biomol. Chem., 2014,12, 7397-7409.



42.Substituted DiphenylButadiynes: a Computational Study of Geometries and Electronic Transitions using DFT/TD-DFT.
A. K.Pati, S. J. Gharpure and A. K. Mishra, Phys. Chem. Chem. Phys.,2014, 16, 14015-14028.



41.Tandem Nucleophilic Addition/Oxa-Michael Reaction for the Synthesis of cis-2,6-DisubstitutedTetrahydropyrans.
S. J. Gharpure, J. V. K. Prasad and KalisankarBera,Eur. J. Org. Chem., 2014,3570-3574.



40. Stereoselective Synthesis of Oxa-Bowls by Nucleophilic Addition to Oxonium Ions: Observation of Nucleophile-Dependent Hydride Migration.
S. J. Gharpure and S. K. Porwal, Eur. J. Org. Chem., 2013, 7277-7281.




39. Coordination Polymers via Self-assembly of Silver(I) and cis-Bisnitrile-oxa-bowl Derivatives.
P. Niranjana, A. Pati, S. K. Porwal, V. Ramkumar, S. J. Gharpure and D. K. Chand, CrystEngComm.,2013.15, 9623-9633.




38. Hetero Diels-Alder Reaction of Olefin with o-Quinone Methides Generated Using (±) Binolphosphoric Acid for the Stereoselective Synthesis of 2,4-Diarylbenzopyrans: Application to the Formal Synthesis of Myristinin B/C.
S. J. Gharpure, A. M. Sathiyanarayananand P. K. Vuram, RSC Adv., 2013,3, 18279-18282.




37. Deciphering the Photophysical Role of Conjugated Diyne in Butadiynyl Fluorophores: Synthesis, Photophysical and Theoretical Study.
A. K. Pati, M. Mohapatra, P. Ghosh, S. J. Gharpure and A. K. Mishra, Phys. Chem. A.,2013, 117, 6548-6560.




36. Stereoselective synthesis of benzoxepines using tandem alkylation-Michael addition to vinylogous carbonates.
S. J. Gharpure and S. R. B. Reddy, Eur. J. Org. Chem., 2013, 2031-2038.




35. Stereoselective Synthesis of Substituted 1,4-Oxazepanes by Intramolecular Reductive Etherification.
S. J. Gharpure and J. V. K. Prasad, Eur. J. Org. Chem., 2013, 2076-2079.




34. Synthesis of Oxa-, Aza- and Thia-Bowls and Cages.
S. J. Gharpure and S. K. Powal, Org. Prep. Proc. Int., 2013, 45, 81. (Invited review).




33. Stereoselective Synthesis of Oxa- and Aza-Angular Triquinanes Using Tandem Radical Cyclization to Vinylogous Carbonates and Carbamates.
S. J. Gharpure, P. Niranjana and S. K. Powal, Org. Lett., 2012, 14, 5476. (Highlighted in Synfacts, 2013, 9(1), 0033).




32. Stereoselective Synthesis and Applications of Nitrogen Substituted Donor-Acceptor Cyclopropanes (N-DACs) in the Divergent Synthesis of Azacycles.
S. J. Gharpure, U. Vijayasree and S. R. B. Reddy, Org. Biomol. Chem., 2012, 10, 1735.




31. Stereoselective Synthesis of C-Substituted Morpholine Derivatives using Reductive Etherification Reaction: Total Synthesis of Chelonin C.
S. J. Gharpure and J. V. K. Prasad, J. Org. Chem., 2011, 76, 10325 .




30. Enantioselective Total Synthesis of (+)-Hagen's Gland Lactones.
S. J. Gharpure, L. N. Nanda, and M. K. Shukla, Eur. J. Org. Chem., 2011, 6632. (Among the top 10 most downloaded paper for October 2011).




29. Stereoselective Synthesis of 2,3-Disubstituted Dihydrobenzofuran using Alkyne Prins Type Cyclization to Vinylogous Carbonates.
S. J. Gharpure, V. Prasath, J. Chem. Sci., 2011, 123, 943. (invited article - International Year of Chemistry) .




28. Stereoselective synthesis of oxazino[4,3-a]indoles employing oxa-Pictet-Spengler reaction of indoles bearing N-tethered vinylogous carbonate.
S. J. Gharpure, A. M. Sathiyanarayanan, Chem. Commun., 2011, 47, 3625.




27. Alkyl radical cyclization to vinylogous carbonates for the stereoselective synthesis of unsymmetrical dioxa-cage compounds: Effect of conformation on the rate of cyclization v/s reduction.
S. J. Gharpure, S. K. Porwal, Tetrahedron, 2011, 67, 1216 .




26. Tandem SN2-Michael Addition to Vinylogous Carbonates for the Stereoselective Construction of 2,3,3,5-Tetrasubstituted Tetrahydrofurans.
S. J. Gharpure, S. R. B. Reddy, Tetrahedron Lett., 2010, 51, 6093.




25. Tandem Radical Cyclization Based Strategy for the Synthesis of Oxa- and Aza-Cages: A Case of Fragmentation v/s Cyclization.
S. J. Gharpure, S. K. Porwal, Tetrahedron Lett., 2010, 51, 3324 .




24. Stereoselective Synthesis of Donor-Acceptor Substituted Cyclopropafuranones by Intramolecular Cyclopropanation of Vinylogous Carbonates: Divergent Synthesis of Tetrahydrofuran-3-one, Tetrahydropyran-3-one and Lactones.
S. J. Gharpure, M. K. Shukla, U. Vijayasree Org. Lett., 2009, 11, 5466.




23. Topologically Driven Tandem Radical Cyclization Based Strategy for the Synthesis of Oxa and Aza-Cages.
S. J. Gharpure, S. K. Porwal, Tetrahedron Lett., 2009, 50, 7162 .




22. Tandem Alkylation-Michael Addition to Vinylogous Carbonates for the Stereoselective Construction of 2,3,3,6-Tetrasubstituted Tetrahydropyrans.
S. J. Gharpure, S. R. B. Reddy, Org. Lett., 2009, 11, 2519.




21. o-Quinone Methide Based Approach to Isoflavans: Application to the Total Syntheses of Equol, 3'-Hydroxyequol and Vestitol.
S. J. Gharpure, A. M. Sathiyanarayanan, P. Jonnalagadda, Tetrahedron Lett., 2008, 49, 2974.




20. Stereoselective Synthesis of New Oxa-Cages via Alkyl Radical Cyclization to Vinylogous Carbonates.
S. J. Gharpure, S. K. Porwal, Synlett, 2008, 242 .




19. Stereoselective Synthesis of 1,2,2-Trisubstituted Indane Derivatives Using Tandem SN2-Michael Addition Sequence.
S. J. Gharpure, S. R. B. Reddy, U. Sanyal, Synlett, 2007, 1889 .





Ph.D and Post-Doctoral Work :


18. An Enantiospecific Strategy to All Four Diastereomers of A-Ring Enyne Synthon of 1 ,25- Dihydroxyvitamin D3.
A. Srikrishna, S. J. Gharpure, P. P. Kumar, Ind. J. Chem. B 2006, 45B, 2736.


17 An Enantiospecific Synthesis of 2-Pupukeanone.
A. Srikrishna, P. R. Kumar, S. J. Gharpure, Ind. J. Chem. B 2006, 45B, 1909.


16. A Central Strategy for Converting Natural Products into Fluorescent Probes.
M. D. Alexander, M. D. Burkart, M. S. Leonard, P. Portonovo, B. Liang, X. Ding, M. M. Joulli, B. M. Gulledge, J. B. Aggen, A. R. Chamberlin, J. Sandler, W. Fenical, J. Cui, S. J. Gharpure, A. Polosukhin, H.-R. Zhang, P. A. Evans, A. D. Richardson, M. K. Harper, C. M. Ireland, B. G. Vong, T. P. Brady, E. A. Theodorakis, J. J. La Clair, Chem. Bio. Chem. 2006, 7, 409.


15. Enantiospecific Synthesis of (+)-2-Thiocyanatoneopupukeanane.
A. Srikrishna, S. J. Gharpure, Proc. of AP Akademi of Sciences 2005, 9, 115.


14. Enantioselective Total Synthesis of the Potent Antitumor Agent (-)-Mucocin using a Temporary Silicon-Tethered (TST) Ring-Closing Metathesis (RCM) Cross-Coupling Reaction.
P. A. Evans, J. Cui, S. J. Gharpure, A. Polosukhin, H. -R. Zhang, J. Am. Chem. Soc. 2003, 125, 14702.


13. Stereoselective Construction of cis-2,6-Disubstituted Tetrahydropyrans via the Reductive Etherification of ?-Trialkylsilyloxy Substituted Ketones: Total Synthesis of (-)-Centrolobine.
P. A. Evans, J. Cui, S. J. Gharpure, Org. Lett. 2003, 5, 3883.


12. Stereoselective Construction of Cyclic Ethers using a Tandem Two-Component Etherification: Elucidation of the Role of Bismuth Tribromide.
P. A. Evans, J. Cui, S. J. Gharpure, R. J. Hinkle, J. Am. Chem. Soc. 2003, 125, 11456.


11. Stereochemistry of the Marine Sesquiterpene 2-Thiocyanatoneopupukeanane: Crystal Structure of Neopupukean-2-yl 4-nitrobenzoate.
A. Srikrishna, S. J. Gharpure, P. Venugopalan, Ind. J. Chem. B 2003, 42B, 129.


10. Chiral Synthons from Carvone. Part 56. Enantiospecific Synthesis of (-)-4-Thiocyanatoneopupukeanane.
A. Srikrishna, S. J. Gharpure, ARKIVOC 2002, 7, 52.


9. A Ring Closing Metathesis Based Approach for the Spiroannulation of Cyclopentanes and Cyclohexanes. Formal Synthesis of (±)-Acorones.
A. Srikrishna, M. S. Rao, S. J. Gharpure, N. C. Babu, Synlett 2001, 1986.


8. Enantiospecific Synthesis of B-seco-C-Aromatic Taxanes.
A. Srikrishna, T. J. Reddy, P. P. Kumar, S. J. Gharpure, Ind. J. Chem. B 2001, 40B, 905.


7. Enantiospecific Total Synthesis of (-)-4-Thiocyanatoneopupukeanane.
A. Srikrishna, S. J. Gharpure, J. Org. Chem. 2001, 66, 4379.


6. An Enantiospecific Synthesis of (-)-2-Pupukeanone via a Rhodium Carbenoid C-H Insertion Reaction.
A. Srikrishna, P. R. Kumar, S. J. Gharpure, Tetrahedron Lett. 2001, 42, 3929.


5. Novel Formation of Chloromethanesulfinates in the Methanesulfonylation Reaction of Hindered Alcohols.
A. Srikrishna, S. J. Gharpure, Synlett 2000, 1354.


4. Enantiospecific Total Synthesis of both Enantiomers of 2-Thiocyanatoneopupukeanane from (R)-Carvone.
A. Srikrishna, S. J. Gharpure, J. Chem. Soc. Perkin Trans. 1 2000, 3191.


3. A Simple, Enantiospecific Approach to both Enantiomers of 1?,25-Dihydroxyvitamin D-3 A-Ring Precursors from (R)-Carvone.
A. Srikrishna, S. J. Gharpure, P. P. Kumar, Tetrahedron Lett. 2000, 41, 3177.


2. Enantiospecific First Total Synthesis of (-)-4-Thiocyanatoneopupukeanane.
A. Srikrishna, S. J. Gharpure, Tetrahedron Lett. 1999, 40, 1035.


1. An Intramolecular Rhodium Carbenoid C-H Insertion Approach to Chiral Isotwistanes. Synthesis of (-)-Neopupukean-4,10-dione and (-)-Neopupukean-10-one.
A. Srikrishna, S. J. Gharpure, Chem. Commun. 1998, 1589.

 

 
 
 
//////